Mankhwala otsutsana ndi kutupa m'magazi amakono amapezeka m'magulu osiyanasiyana - onse opangidwa ndi ufa, ndi mapiritsi, ndi majekeseni, ndipo, ndithudi, mwa mawonekedwe a mafuta ndi mafuta. Mmodzi mwa ma NSAID wotchuka kwambiri monga mawonekedwe a gel osatchedwa Diclofenac. Izi ndi chifukwa cha zinthu zingapo: poyamba, mankhwalawa alibe mtengo wapatali, ndipo kachiwiri, ndi othandiza kwambiri, ndipo katatu, kutchuka kwa dzina la mankhwala kumathandizidwa ndi mitundu ina - jekeseni ndi mapiritsi omwewo.
Kupanga gel Diclofenac
Diclofenac imatha kuyimira anti-inflammatory os-steroid agent ndipo imakhala ndi gel kuchokera ku diclofenac sodium.
Zothandizira zothandizira gel kuti zilowerere bwino mu matenda ndi kusunga katundu wawo kwa nthawi yaitali ndi izi:
- kukonzedwa kwa ethanol;
- propylene glycol;
- katemera;
- chotsitsa;
- methyl lauryl hydroxybenzonate;
- mafuta a lavender;
- madzi oyera.
Kutulutsa mawonekedwe ndi kusungunuka kwa gel Diclofenac
Gel Diclofenac imapezeka m'mabotolo a aluminium kwa 50 ndi 40 g.
Kuphatikiza pa voliyumu, chiwerengero cha zinthuzo chimasiyananso:
- Gelisi ya Diclofenac 5% - pa 1 g yalemera imakhala 50 mg ya sodium ya diclofenac;
- Diclofenac gel 3% - 1 g ya gel osakaniza 30 mg ya diclofenac sodium;
- Dellofenac gel 1% - 1 g ya gel osakaniza ndi 10 mg wothandizira kwambiri - diclofenac sodium.
Mafuta a Diclofenac palibe, koma gel ndilo lokha.
Mankhwala a gel Diclofenac
Diclofenac ndi mankhwala omwe amachititsa kuti mankhwalawa asokonezeke, komanso amatchedwa anti-inflammatory properties. Zimaletsa mavitamini COX-2 ndi COX-1, komanso zimasokoneza kaphatikizidwe ka arachidonic asidi ndi metabolism ya prostaglandins, yomwe imapanga chingwe cha kutupa. Choncho, gelisi imathetsa kufalikira kwa kutukusira, komanso imalepheretsa chitukuko chake m'matumba ozungulira.
Chifukwa cha zidazi, Diclofenac imagwiritsidwa ntchito ngati decongestant ngati kutupa kumachitika ndi kutupa. Amaperekedwanso kuti azitha kupwetekedwa ngati kupweteka kwapanyumba kumalo ngati kupweteka kumayambitsa ndondomeko yotupa.
Diclofenac imachepetsa kutupa m'magawo otsekemera, kutontholetsa kuuma. Komanso m'madera otupa, amathetsa ululu, kapena amachepetsa kwambiri.
Diclofenac gel malangizo
Malangizo ogwiritsira ntchito Gel Diclofenac 5%, komanso 3% ndi 1% si osiyana. Kusiyana kumeneku kumakhala ndi mphamvu yogwira ntchito, ndipo cholinga chake chimadalira kukula kwa zizindikiro. Mwachitsanzo, gelisi la Diclofenac liri ndi mphamvu ya 5% yogwiritsidwa ntchito popweteka kwambiri mu rheumatism .
Zizindikiro zogwiritsira ntchito gel Diclofenac
Diclofenac akulamulidwa ku matenda awa:
- rheumatic pathologies - bursitis , tendovaginitis, etc ;;
- Kupweteka kwa minofu kumbuyo kwa rheumatism kapena kuwonongeka kwa minofu ya minofu;
- Kuthamanga kwa ziwalo pambuyo pake.
Gelisi ya Diclofenac imagwiritsidwa ntchito kunja, ndipo chiwerengero cha osagwiritsa ntchito chimadalira kukula kwa dera lopweteka.
Komabe, pali zifukwa zambiri zomwe zimagwiritsidwa ntchito pogwiritsa ntchito gel osakaniza:
- Diclofenac gel 1% - ntchito imodzi - mpaka 4 g;
- Diclofenac gel 3% - ntchito imodzi - mpaka 3 g;
- Diclofenac gel 5% - osagwiritsa ntchito mpaka 2 g.
Ana omwe ali ndi zaka zoposa 12 komanso akuluakulu amalimbikitsidwa kugwiritsa ntchito gel 3-4 patsiku ndi kusinthasintha.
Zotsutsana ndi kugwiritsa ntchito gel Diclofenac
Diclofenac sichitha kugwiritsidwa ntchito pazinthu zotsatirazi:
- mimba (malingaliro 3 trimester);
- lactation;
- zaka za ana (mpaka zaka 6);
- mabala, kuyaka;
- mankhwala osokoneza bongo kapena asthma omwe amayamba chifukwa cha kugwiritsa ntchito mankhwala osagwiritsa ntchito mankhwala oletsa kutupa.
Ngati pali matenda a magazi, Gel Diclofenac 5% ayenera kugwiritsidwa ntchito mosamala.