Diclofenac analogues

Diclofenac ndi gulu la mankhwala omwe amagwiritsidwa ntchito pa matenda osiyanasiyana opweteka a m'maganizo ndi minofu. Mankhwalawa amatanthauza mankhwala osagwiritsa ntchito mankhwala omwe amatsutsana kwambiri ndi zotsatira zake. Pankhani imeneyi, nthawi zambiri pamakhala kofunika kupeza analoji - ogwira ntchito komanso nthawi yomweyo. Komanso, sizingatheke koma kunena kuti asayansi ochokera ku UK adafuna kuchotsa Diclofenac chifukwa, malinga ndi maphunziro awo, amachititsa kuti chiopsezo cha mtima chiwonjezeke, chomwe lero ndi chimodzi mwa "zikwapu" zazikulu za anthu. Kuitana kumeneku sikungakhudze madokotala a pakhomo, ndipo Diclofenac akadakalipira kuti adziwe mankhwala.

Kenaka, tiyang'ana mankhwala omwe angathe kutenga Diclofenac.

Diclofenac Analogs mu Majekesero ndi Zowona Zambiri

Mankhwala a diclofenac mu jekeseni si ovuta kupeza, ngati inu mukuyang'ana mfundo ya chinthu chomwecho chogwira ntchito. Sodium ya Diclofenac ili mu Voltaren, Diklak, Almiral, ndi ena.

Ndikovuta kwambiri kupeza wothandizira ofanana ndi chinthu china chogwira ntchito. Iye ndi Arthrosan - ntchito yake yaikulu - meloxicam. Ndiyo njira yosankha yokha ya COX-2, yomwe imayimiranso mankhwala osagwiritsidwa ntchito poletsa kutupa, omwe amakhala ndi 89%. N'zochititsa chidwi kuti Diclofenac, malinga ndi malangizo, amaloledwa kugwiritsidwa ntchito panthawi yomwe ali ndi pakati, ngati ntchito yake imadziwonetsera yokhazokha chifukwa cha chiopsezo kwa mwana ndi mayi, ndipo, panthaƔi imodzimodziyo, Arthrosan imatsutsana kwambiri ndi mimba.

Motero, tinganene kuti Diclofenac ndi njira yatsopano yamakono komanso yothetsera mavuto, ngakhale chenjezo la asayansi a ku Britain. Arthrosan imakhala ndi zotsatira zambiri kuchokera ku machitidwe onse a thupi.

Dalolofenac ya Analog mu maonekedwe a meloxicam sayenera kugwiritsidwa ntchito kwa nthawi yaitali.

Diklofenac yamakono yamakono ndi Naproxen. Amaperekedwa mwa mawonekedwe a jekeseni, gels ndi mapiritsi, ali ndi mphamvu yochepa kuposa diclofenac sodium, koma nthawi yomweyo ndi mankhwala oopsa.

Naproxen imatanthawuza panthawi yomweyo magulu asanu a mankhwala:

Mankhwala ena odana ndi kutupa omwe angathe kutenga Diclofenac ndi Ibuprofen. Ndipotu ichi ndi chiganizo chake ngati tiyerekezera zotsatira zake, zotsutsana ndi zizindikiro. Ibuprofen ndizochokera ku phenylpropionic acid, ndipo, monga zina za NSAID, zimalepheretsa COX.

Mafotokozedwe a Diclofenac m'mapiritsi

Zizindikiro za Diclofenac m'mapiritsi, kuphatikiza pa ndalama zomwe tazitchulazi, ndi:

Tiyenera kukumbukira kuti Sulindack sichimavulaza kwambiri mmimba kuposa Indomethacin, koma nthawi yomweyo imakhala yoopsa kwa chiwindi.

Mafotokozedwe a mafuta a diclofenac

Mafuta otetezedwa kwambiri pakati pa mafananidwe a Diclofenac ndi Clofezon. Phenylbutazone imalekerera kwambiri, koma imatha kupitirira aspirin. Indomethacin ndi mankhwala amphamvu kwambiri omwe sali ndi steroidal anti-inflammatory drug, ndipo motero amauzidwa nthawi zambiri, pamene akuwononga kwambiri thupi.

Diclofenac gel analogues

Zamphamvu kwambiri pakati pa gels ndi Piroxicam ndi Ketoprofen. Ambiri ogwiritsidwa ntchito naproxen amachokera kufooka kuchita ndi zovulaza thupi.

Makandulo a makandulo Fufuzani Magulu Mayiko Uzani-anzanu Buku la alendo Mbiri yathu Perekani Chithandizo

Indomethacin ndi mankhwala ogwiritsidwa ntchito kwambiri pa gululi, choncho sizingavomerezedwe kuigwiritsa ntchito nthawi zonse.